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authFullName_s : Sébastien Papot
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Monitoring glycosidase activity for clustered sugar substrates, a study on β-glucuronidase

Yoan Brissonnet , Guillaume Compain , Brigitte Renoux , Eva-Maria Krammer , Franck Daligault , et al.
RSC Advances, 2019, 9 (69), pp.40263-40267. ⟨10.1039/c9ra08847d⟩
Journal articles hal-02992513v1

Evaluation of Cytotoxic Properties of a Cyclopamine Glucuronide Prodrug in Rat Glioblastoma Cells and Tumors

Souheyla Bensalma , Corinne Chadeneau , Thibaut Legigan , Brigitte Renoux , Afsaneh Gaillard , et al.
Journal of Molecular Neuroscience, 2015, 55 (1), pp.51-61. ⟨10.1007/s12031-014-0395-3⟩
Journal articles hal-01328060v1
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Absolute configuration of a [1]rotaxane determined from vibrational and electronic circular dichroism spectra

Andrew R Puente , Adrien Bessaguet , Noël Pairault , Grégory Pieters , Jeanne Crassous , et al.
Chirality, 2021, 33 (11), pp.773-782. ⟨10.1002/chir.23365⟩
Journal articles hal-03360296v1
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Surface functionalization by covalent immobilization of an innovative carvacrol derivative to avoid fungal biofilm formation

Aïcha Gharbi , Thibaut Legigan , Vincent Humblot , Sébastien Papot , Jean-Marc Berjeaud
AMB Express, 2015, 5 (1), pp.9. ⟨10.1186/s13568-014-0091-2⟩
Journal articles hal-01143973v1

A self-immolative dendritic glucuronide prodrug of doxorubicin

Marion Grinda , J. Clarhaut , Brigitte Renoux , Isabelle Tranoy-Opalinski , Sébastien Papot
MedChemComm, 2012, 3 (1), pp.68-70. ⟨10.1039/c1md00193k⟩
Journal articles hal-00682705v1
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NDMA formation mechanism by chloramination of tertiary amines

Julien Le Roux , Hervé Gallard , Jean-Philippe Croué , Sébastien Papot , Marie Deborde
2012 AWWA Water Quality Technology Conference & Exposition, Nov 2012, Toronto, Canada
Conference papers hal-01211527v1

2-Acetamido-2-deoxy- l -iminosugar C -Alkyl and C -Aryl Glycosides: Synthesis and Glycosidase Inhibition

Balkis Eddhif , Justin Lange , Nadia Guignard , Yann Batonneau , Jonathan A. Clarhaut , et al.
European Journal of Organic Chemistry, 2018, 2018 (40), pp.5477-5488. ⟨10.1002/ejoc.201800678⟩
Journal articles hal-02172201v1

In situ targeted activation of an anticancer agent using ultrasound-triggered release of composite droplets

Sergii Kolodych , Chloé Michel , Sébastien Delacroix , Oleksandr Koniev , Anthony Ehkirch , et al.
European Journal of Medicinal Chemistry, 2017, 142, pp.2-7. ⟨10.1016/j.ejmech.2017.03.057⟩
Journal articles hal-02174984v1
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A dendritic β-galactosidase-responsive folate–monomethylauristatin E conjugate

Jérôme Alsarraf , Elodie Peraudeau , Pauline Poinot , I. Tranoy-Opalinski , Jonathan Clarhaut , et al.
Chemical Communications, 2015, 51 (87), pp.15792-15795. ⟨10.1039/C5CC05294G⟩
Journal articles hal-03127679v1
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Enzyme‐Cleavable Linkers for Protein Chemical Synthesis through Solid‐Phase Ligations

Skander A Abboud , Mehdi Amoura , J.B Madinier , Brigitte Renoux , Sébastien Papot , et al.
Angewandte Chemie International Edition, 2021, 60 (34), pp.18612-18618. ⟨10.1002/anie.202103768⟩
Journal articles hal-03335485v1
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Diastereoselective synthesis of [1]rotaxanes via an active metal template strategy

Noël Pairault , Adrien Bessaguet , Romain Barat , Lucas Frédéric , Grégory Pieters , et al.
Chemical Science, 2021, 12 (7), pp.2521-2526. ⟨10.1039/d0sc05369d⟩
Journal articles hal-03105942v1
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Design, synthesis and biological evaluation of quinoline-2-carbonitrile-based hydroxamic acids as dual tubulin polymerization and histone deacetylases inhibitors

Camille Hauguel , Sarah Ducellier , Olivier Provot , Nada Ibrahim , Diana Lamaa , et al.
European Journal of Medicinal Chemistry, 2022, 240, pp.114573. ⟨10.1016/j.ejmech.2022.114573⟩
Journal articles hal-03752715v1

Etude de l’effet du premier vecteur glucuronylé de la cyclopamine sur les cellules initiatrices de glioblastomes

Anais Balbous , Brigitte Renoux , Ulrich Cortes , Serge Milin , Karline Guilloteau , et al.
6ème journée de la Recherche Tours-Poitiers, Nov 2013, Poitiers, France
Conference poster hal-02538758v1

Impact of operation conditions, foulant adsorption, and chemical cleaning on the nanomechanical properties of ultrafiltration hollow fiber membranes

Audrey Allavena , Sylvie Liu , Thomas Ribette , Ninette Abou Mrad , Thierry Chiavassa , et al.
Colloids and Surfaces A: Physicochemical and Engineering Aspects, 2018, 549, pp.34-42. ⟨10.1016/j.colsurfa.2018.04.003⟩
Journal articles hal-02121394v1
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Erratum to: Surface functionalization by covalent immobilization of an innovative carvacrol derivative to avoid fungal biofilm formation

Aïcha Gharbi , Thibaut Legigan , Vincent Humblot , Sébastien Papot , Christine Imbert , et al.
AMB Express, 2015, 5 (1), pp.56. ⟨10.1186/s13568-015-0141-4⟩
Journal articles hal-01206241v1
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The Lossen rearrangement from free hydroxamic acids

Mikaël Thomas , Jérôme Alsarraf , Nahla Araji , Isabelle Tranoy-Opalinski , Brigitte Renoux , et al.
Organic & Biomolecular Chemistry, 2019, 17 (22), pp.5420-5427. ⟨10.1039/c9ob00789j⟩
Journal articles hal-02380109v1
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Cell–cell interactions via non-covalent click chemistry

Chad Plumet , Achmet Said Mohamed , Tanguy Vendeuvre , Brigitte Renoux , Jonathan Clarhaut , et al.
Chemical Science, 2021, 12 (26), pp.9017-9021. ⟨10.1039/D1SC01637G⟩
Journal articles hal-03285569v1

Development and evaluation of β-galactosidase-sensitive antibody-drug conjugates

Sergii Kolodych , Chloé Michel , Sébastien Delacroix , Oleksandr Koniev , Anthony Ehkirch , et al.
European Journal of Medicinal Chemistry, 2017, 142, pp.376 - 382. ⟨10.1016/j.ejmech.2017.08.008⟩
Journal articles hal-01649358v1

Reduction–rebridging strategy for the preparation of ADPN-based antibody–drug conjugates

Oleksandr Koniev , Igor Dovgan , Brigitte Renoux , Anthony Ehkirch , Jitka Eberova , et al.
MedChemComm, 2018, 9 (5), pp.827-830. ⟨10.1039/C8MD00141C⟩
Journal articles hal-02169901v1
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A Novel Proteomics-Based Strategy for the Investigation of Peptide Sequences in Extraterrestrial Samples

Justin Lange , Fabiola Djago , Balkis Eddhif , Quentin Remaury , Alexander Ruf , et al.
Journal of Proteome Research, 2020, 20 (2), pp.1444-1450. ⟨10.1021/acs.jproteome.0c00700⟩
Journal articles hal-03052767v1

Synthesis and Antitumor Efficacy of a β-Glucuronidase-Responsive Albumin-Binding Prodrug of Doxorubicin.

Thibaut Legigan , Jonathan Clarhaut , Brigitte Renoux , Isabelle Tranoy-Opalinski , Arnaud Monvoisin , et al.
Journal of Medicinal Chemistry, 2012, 55 (9), pp.4516-20. ⟨10.1021/jm300348r⟩
Journal articles hal-00710692v1
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Rotaxane-based architectures for biological applications

Noël Pairault , Romain Barat , I. Tranoy-Opalinski , Brigitte Renoux , Mikaël Thomas , et al.
Comptes Rendus. Chimie, 2016, 19 (1-2), pp.103-112. ⟨10.1016/j.crci.2015.05.012⟩
Journal articles hal-03127619v1
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A mechanically interlocked molecular system programmed for the delivery of an anticancer drug

Romain Barat , Thibaut Legigan , I. Tranoy-Opalinski , Brigitte Renoux , Elodie Peraudeau , et al.
Chemical Science, 2015, 6 (4), pp.2608-2613. ⟨10.1039/c5sc00648a⟩
Journal articles hal-03127729v1
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Stimuli‐Responsive Metal Complexes for Biomedical Applications

Ivanna Amarsy , Sébastien Papot , Gilles Gasser
Angewandte Chemie International Edition, 2022, 61 (40), pp.e202205900. ⟨10.1002/anie.202205900⟩
Journal articles hal-03713992v1
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A β-Cyclodextrin-Albumin Conjugate for Enhancing Therapeutic Efficacy of Cytotoxic Drugs

Chad Plumet , Rémi Châtre , Fabiola Djago , Elodie Péraudeau , Quentin Blancart-Remaury , et al.
Bioconjugate Chemistry, 2022, 33 (6), pp.1138-1144. ⟨10.1021/acs.bioconjchem.2c00182⟩
Journal articles hal-03765739v1
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NDMA Formation by Chloramination of Ranitidine: Kinetics and Mechanism

Julien Le Roux , Hervé Gallard , Jean-Philippe Croué , Sébastien Papot , Marie Deborde
Environmental Science and Technology, 2012, 46 (20), ⟨10.1021/es3023094⟩
Journal articles hal-01201597v1

Targeting the tumour microenvironment with an enzyme-responsive drug delivery system for the efficient therapy of breast and pancreatic cancers

Brigitte Renoux , Florian Raes , Thibaut Legigan , Elodie Péraudeau , Balkis Eddhif , et al.
Chemical Science, 2017, 8 (5), pp.3427-3433. ⟨10.1039/C7SC00472A⟩
Journal articles hal-02174996v1

A β-glucuronidase-responsive albumin-binding prodrug for potential selective kinase inhibitor-based cancer chemotherapy

Guillaume Compain , Nassima Oumata , Jonathan A. Clarhaut , Elodie Péraudeau , Brigitte Renoux , et al.
European Journal of Medicinal Chemistry, 2018, 158, pp.1-6. ⟨10.1016/j.ejmech.2018.08.100⟩
Journal articles hal-02169782v1
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A galactosidase-responsive doxorubicin-folate conjugate for selective targeting of acute myelogenous leukemia blasts

Jonathan Clarhaut , Sylvain Fraineau , Joëlle Guilhot , Elodie Péraudeau , Isabelle Tranoy-Opalinski , et al.
Leukemia Research, 2013, 37 (8), pp.948 - 955. ⟨10.1016/j.leukres.2013.04.026⟩
Journal articles inserm-02444614v1
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Induced-volatolomics for the design of tumour activated therapy

Rémi Châtre , Estelle Blochouse , Rony Eid , Fabiola Djago , Justin Lange , et al.
Chemical Science, 2023, 14 (18), pp.4697-4703. ⟨10.1039/d2sc06797h⟩
Journal articles hal-04098727v1